*Please inquire the availability for this product. Azamulin is a semi-synthetic pleuromutilin prepared by sequential reaction of dihydropleuromutilin tosylate with 2-amino-1,2,4-triazole-5-thiol. While azamulin is a broad spectrum antibiotic in the pleuromutilin class, this aspect of its bioprofile has received little attention. In fact, the triazole substituent added to nominally improve the drug's bioavailability, imparted an unusual selectivity for the inhibition of specific cytochrome P450 mixed function oxidase sub-types, important for understanding the manner in which the body metabolises drugs or xenobiotics.

Additional Information

Synonyms	TMD 85-530, SA 85530b
Product #	A-2663
CAS #	76530-44-4
Formula	C24H36N4O4S
MW	476.6
Appearance	White solid
Purity	>99% by HPLC
Solubility	Soluble in DMSO and Methanol
Melting Point	>128°C
Storage Temp	-20°C
Therapeutic Area	Infectious Diseases
Use	Azamulin is a broad spectrum antibiotic

Additional Information

MDL Number	MFCD00865055
InChI	InChI=1S/C24H38N4O4S/c1-6-22(4)11-16(32-17(30)12-33-21-26-20(25)27-28-21)23(5)13(2)7-9-24(14(3)19(22)31)10-8-15(29)18(23)24/h13-14,16,18-19,31H,6-12H2,1-5H3,(H3,25,26,27,28)/t13-,14+,16-,18+,19+,22-,23?,24+/m1/s1
SMILES	CC[C@@]1(C[C@H](C2([C@@H](CC[C@@]3([C@H]2C(=O)CC3)[C@H]([C@@H]1O)C)C)C)OC(=O)CSc4[nH]c(nn4)N)C